Golovinsky – List of selected publications

A. Spassov, E. Golovinsky, G. Russev - "Oxydative Cyclisierung von Arylidenamidrazonen zu 2,4,5-triarylsubstituierten 1,2,4-Triazolonen" - Chem. Ber. 96 (11), (1963) 1996.

A. Spassov, E. Golovinsky, G. Demirov - "Umsetzung von Amidrazonen mit Chlorameisensaureathylester. Darstellung 3,4-Diarylsubstituituerten 1,2,3-Triazolonen-(5)" - Chem. Ber. 98 (3), (1965) 932.

K. Markov, E. Golovinsky - "Chemische Konstitution und antibakterielle Aktivitat der Pyridincarbonsaure-Thioanilide" - Naturwissenschaften 47 (9), (1960) 450.

E. Golovinsky, K. Markov - "Die Wirkung des Nikotinsaurenitrils und -amidoxims als Wachstumsfaktoren fur Bact. Proteus Vulg. und Staphylococcus aureus" - Z. Naturforsch. 138 (11), (1958) 725.

K. Markov, E. Golovinsky - "Biologische Eigenschafften eines gegen Nikotinsaurethioanilid resistenten B. Proteus vulgaris-Stammes" - Z.Naturforsch. 16b (4), (1961) 258.

K. Markov, G. Saev, E. Golovinsky - "Adaptive chain in the Conversion of Antimetabolites into Metabolites" - Nature (London) 187 n 4742, (1960) 1041.

W. Ivanov, K. Markov, E. Golovinsky, T. Charisanova - "Die Bedeutung der Oberflechen-Lipide fur einige biologische Eigenschaften eines Ps. Aeroginosa-Stammes" - Z. Naturforsch. 198 (7), (1964) 604.

D. Paskov, A. Spassov, I. Krushkov, E. Golovinsky - "Structure-Activity Relationship of Pyridine Derivatives" - Arch. Intern. Pharmac. Therap. 157 (1965) 132.

E. Golovinsky, S. Pantcheva-Golovinsky, H. M. Rauen - "Der Wirkungsmechanismus von Thiopicolinsaureamid bei Neurospora crassa" - Arzneimittel-Forsch. 18 (1968) 1232.

H. M. Rauen, K. Norpoth, E. Golovinsky - "Direkte Hydroxylierung von Endoxan" - Naturvissenschaften 54 (1968) 589.

H. M. Rauen, E. Golovinsky, K. Norpoth - "Die elekrophoretische Beweglichkeit von Rattenblut-Erytrocyten nach Zufuhr von Endoxan ober NH-Lost" - Klinische Wochenschr. 46 (1968) 276.

E. Golovisky - "Uber das Verhalten eineiger Orotsaure-Analoga und -Derivate unter den Bedingungen der Tsuji-Reaktion" - Z. Chemie 8 (1968) 421.

A. Spassov, E. Golovinsky, G. Russev - "Synthese von s-Tetrazolo-(1,5-A)- und 2-(Pyrazolyl-1)-uracile" - Z. Chemie 8 (1968) 421.

A. Spassov, E. Golovinsky, G. Russev - "Uber die Umsetzung von Amidrazonen mit Я-Diketonen und β-Ketoestern" - Chem. Ber. 99 (1968) 3728.

A. Spassov, E. Golovinsky, G. Demirov - "Umsetzung von Amidrazonen mit Ameisensaure-Aethylester. Darstellung von 3,4-diarylsubstituierten 1,2,4-Triazolonen-(5)" - Chem. Ber. 99 (1966).3734.

E. Golovinsky, A. Spassov, E. Roussinova - "Die Wirkung eineiger Orotaldehyd - Derivate als Orotsaurentagonisten bei Neurospora crassa" - Z. Naturforschg. 24b (10), (1969) 1315.

I. Kaneti, E. Golovinssky, I. Yukhnovsky, D. Genchev - "A Study of Some Orotic Acid Derivatives and Analogues by Huckel's Method of Molecular Orbital. I.Active Site by Orotidine-5'-Phosphate-Pyrophosphorylase" - J. Theor. Biol. 26 (1970) 19.

E. Golovinssky, I. Kaneti, I. Yukhnovsky, D. Genchev - "A Study of Some Orotic Acid Derivatives and Analogues by Huckel's Method of Molecular Orbitals. II.Analogues of the Orotic Acid in the Reaction with Phosphoribosyl-Pyrophosphorylase" - J. Theor. Biol. 26  (1970) 29.

K. Norpoth, E. Golovinsky, H. M. Rauen - "Untersuchungen an hypothetischen Metaboliten des Cyclophosphamids" - Hoppe-Seyler's Z. Physiol. Chem. 351 (1970) 377.

K. Chelbova, E. Golovinsky, A. A. Hadjiolov - "The Action of Some Orotic Acids Analogues on the in vitro Incorporation of ¹⁴C-Orotate into Pyrimidine Nucleotides" - Biochem. Pharmacol. 19 (1970) 2785.

E. Emanuilov, E. Golovinsky - "Heterotransplantation of Ehrlich Ascites Tumor Cells in Rats Pre-Treated with Cytostatics and Antimetabolites" - Z. Naturforschg. 25b (1970) 1175.

J. Kaneti, E. Golovinsky - "Quantitative Relationship between the Electronic Structure and Biological Activity of some Analogues of Orotic Acid" - Chem.-Biol. Interactions 3 (1971) 421.

E. Golovinsky - "Biochemie der Orotsaureantimetabolite" - Hippokrates 43 (1972) 101.

E. Golovinsky - "Zum Wirkungsmechanismus von Orotsaureanaloga" - Studia Biophysica 31/32 (1972) 427.

J. Kaneti, E. Golovinsky, S. Dimova - "A Molecular Orbital Approach to the Study of Some Stages of Purine Metabolic Pathways" - FEBS Symp. 22 (1972) 163-176.

A. Spassov, E. Golovinsky, N. Spassovska, L. Maneva - "Effect of Thio- and Hydrazino-derivatives of Uracil, 6-Azauracil and 6-Azathymine on the Growth of Some Microorganisms in vitro" - Z. Naturforschung 27b (1972) 818.

P.Popov, S. Kavrakirova, I. Belokonsky, E. Golovinsky - "The effect of some cytostatics on tyrosine aminotranspherase activity in rat liver" - Acta Biol. Med. Germ. 29 (1972) 751.

B. Alexiev, S. Stoev, A. Spassov, L. Maneva, E. Golovinsky - "Synthesis and Antibacterial Activity of peptides containing cysteinesulfonamide and its derivatives" - "Peptides 1972", p.245, Elsevier 1973.

K. Hadjiolova, E. Golovinsky, A. A. Hadjiolov - "The site of action of 5-Fluoroorotic acid on the maturation of mouse liver ribonuckeic acids" - Biochim. Biophys. Acta 319, (1973) 375.

E. Golovinsky, E. Emanuilov, N. Spassovska, A. Spassov - "Antitumor effect of 2-thio-4-hydrazinouracil on transplantable tumors" - Neoplasma 22 (1975) 255.

M. Spassova, G. Russev, E. Golovinsky - "Some pyrazoles as inhibitors on purine biosynthesis de novo" - Biochem. Pharmacol. 25  (1975) 923.

E. Golovinsky, L. Maneva, I. Angelov, K. Veljanova, D. Sniker, E. Stankevich - "Antibactetial and antitumor activity of some derivatives of ureidosuccinic acid" - Neoplasma 23 (1976) 43.

H.-E. Jacob, E. Golovinsky, D. Hradecna, G. Lober, L. Maneva – “The effect of Base-analogues present in the growth medium on UV-sensibility of bacteria" - in "Design and mechanism of action of antimetabolites", Varna 1975, Publ. House of BAS, Sofia 1976.

M. Spassova, E. Golovinsky - "Synthesis, structure and antibacterial activity of some alkyltriazenopyrazoles" - Arzneimittel-Forsch. 27 (I), (1977) 758.

E. Golovinsky, B. Alexiev, A. Spassov, S. Stoev, E. Emanuilov, I. Angelov, L. Maneva, Ts. Stoychev - "A new substance effective against transplantable tumors in vivo: L-Cystine-bis-(N,N-β-chloroethyl)-hydrazide" - Neoplasma 24 (1977) 401.

L. Maneva, S. Stoev, B. Alexiev, E. Golovinsky - "Antibakterielle Aktivitat einiger substituirten Cysteinsulfonamide und cysteinsulfonamidhaltiger Peptide" - Pharmazie 34 (1979) 423.

M. Spassova, K. Grantcharov, R. Zakharieva, E. Golovinsky - "Mechnism of Inhibitory Effect of some Pyrazole Derivatives on Purine Biosynthesis de novo" - Biochem. Pharmacol. 29 (1980) 163.

M. Spassova, R. Zakharieva, E. Golovinsky - "Synthese von Diamino- und Trichlormethylaminoderivaten der Pyrazolcarbonsaure" - Z. Chemie 20 (1980) 95.

M. Karaivanova, S. Zakhariev, E. Golovinsky - "Antitumor Effect of N_α-Benzyloxycarbonyl-N,N-bis-(2-halogenoethyl)-Hydrazide Derivatives of Amino Acids" - Neoplasma 27 (2), (1980) 137.

E. Golovinsky "Mutagenic and Carcinogenic Effects of Antimetabolites. In "Short-Texm Systems for Detecting Carcinogene" - K. Norpoth, R. Garner Eds, Springer-Verlag, Berlin-Heidelberg-New York, 1980.

D. Veljanov, A. Rutkov, T. Radoutcheva, D. Harbov, E. Golovinsky - "Influence of D,L-Ureidosuccinic Acid Dihydrazide on some Bioligical Properties of Pseudomonas pseudomallei and of Salmonella typhimurium" - Zbl. Bakt. Hyg. I. Abt. Orig. A 247, (1980) 64.

E. Golovinsky, A. Galabov, E. Stankevich, A. Karparov, L. Maneva, K. Grancharov, N. Chakova, D. Sniker, I. Angelov, E. Velichkova, V. Karabasheva - "Antiviral, Antibacterial and Antitumor Activity of the Hydrazide and the Ethyl Esther of 2,2'-Anhydro-1-(β-D-arabinofuranosyl)-orotic acid" - Arzneimittel-Forschg 30 (II) (12), (1980) 2087.

E. Raikova, D. Gruev, E. Golovinsky - "In vivo Investigation of some Metabolic Changes of 3-[Bis-(2-Chloroethyl)-carbohydrazide]-2,2,5,5-tetramethylpyroline-1-oxyl by  the NBP-Reaktion and ESR-Method" - Biochem. Pharmacol. 30 (1981) 289.

E. Golovinsky, M. Spassova - "Analogs of Pyrimidine and Purine Mononucleotide Precursors as Metabolic Inhibitors" - Pharmac. Therap. 13 (1981) 385.

B. Aleksiev, S. Stoev, S. Zakhariev, E. Golovinsky - "Verwendung von alkalischer Protease des Bacillus subtilis Stammes DY zur Hydrolyse von Aminosauren und Peptidester" - Hoppe Seyler's Z. Physiol. Chem. 362 (1981) 1323.

P. Bontchev, M. Boneva, D. Mehandjiev, E. Golovinsky - "Copper (II) complexes of Hydrazides" - J. Inorg. Nucl. Chem. 43 (3), (1981) 3163.

S. Zakhariev, R. Zakharieva, W. Gryc, S. Stoev, B. Tomicka, E. Golovinsky, B. Alexiev, M. Karaivanova, G. Kupryszewski -  "Derivatives of (R)-2-Amino-3-sulfamoilpropanoic acid" - Polish J. Chemistry 55 (1981) 799.

E. Golovinsky, G. Karamanov, N. Spassovska, L. Maneva, A. Spassov - "Synthese, antibakterielle und geschwulsthemmende Wirkung einie Methylhydrazoniumsalze von Pyrimidinbasen und deren Analoga" - Die Pharmazie 37 (1982) 355.

D. Veljanov, T. Radoutcheva, V. Kantardjiev, E. Stankevich, E. Golovinsky - "Biological Effect  of D,L-Ureidosuccinic acid dihydrazide on Pseudomonas Pseudomallei and Salmonella Typimurium" - Arch. Roum. Path. Exp. Microbiol. 42 (2), (1982) 99.

E. Raikova, D. Kafalieva, I. Ivanov, S. Zakhariev, E. Golovinsky - "EPR study on the interaction on spin-labelled hydrazine mustard derivatives with DNA" - Biochem. Pharmacology 32 (4), (1983) 587.

E. Golovinnsky, K.Norpoth, E. Stankevich, E. Mohtashmpir - "Mutagenicity of hydrazides of pyrimidinenucleotide-precursors in the Salmonella Oxygenase test" - Cancer Letters 19 (1983) 67.

M. Spassova, R. Zakharieva, E. Golovinsky - "Synthese und Strukturaufklarung von Diazonium-derivaten einiger Pyrazole” - Z. Chemie 23 (1983) 295.

N. Spassovska, K. Grancharov, L. Maneva, T. Popov, M. Spassovski, E. Golovinsky, R. Tzanev - "Antibacterial and Antitumor Activity of a Spermine Platinum Complex (II)" - Proc. 13 Int. Congr. Chemotherapy, Vienna 1983, PP. 100-103.

D. Veljanov, T. Radoutcheva, D. Harbov, I. Stankova-Shinderova, E. Stankevich, E. Golovinnsky - "Biological Effect of L-Asparagin Acid Hydrazide on Salmonella Pseudomallei and Salmonella Typimurium"  - Arch. Roum. Path. Exp. Microbiol. 42 (2-3), (1983) 131.

G.-J. Krauss, K. Grancharov, D. Genchev, R. Walther, N. Spassovska, G. Karamanov, H. Reinbothe, E. Golovinsky - "Metabolic Conversion of Orotic Acid Hydrazide into a Nucleotide in Mouse and Rat liver" - Biomed. Biochim. Acta 42 (1983) 1045.

H. Jacob. E. Golovinsky - "Wirkungen von 5-Bromuracil und 5-Bromdesoxyuridine in Kombination mit 8-Azaadenin auf die UV-Empfindlichkeit von Bacterien" - Z. f. Allg. Microbiologie 23 (1983) 495.

R. Pelova, N. Spassovska, L. Maneva, E. Golovinsky - "Synthesis and Biological Activity of Hydrazinopyrimidines with Carbonyl Compounds" - Pharmazie 39 (4), (1984) 270.

N. Spassovska, R. Pelova, L. Maneva, E. Golovinsky - "Synthesis of Platinum Complexes of Glioxal and Pyruvic Acid Thiosemicarbazones" - Pharmazie 39 (4), (1984) 346.

R. Zakharieva, M. Spassova, M. Karaivanova, E. Golovinsky - "Synthesis and Antitumor Activity of Alkyltriazenopyrazoles" - Arzneimittel-Forschg 34 (I) (1984) 6,661-663.

M. Spassova, K. Grancharov, E. Golovinsky - "Cyanopyrazoles as analogs of Purine precursors. I.Inhibotory effect on purine biosynthesis de novo" - Int. J. Biochemystry 16 (10), (1984) 1091.

M. Spassova, E. Golovinsky - "Pharmacobiochemistry of Arylalkyltriazenes and their Application in Cancer Chemotherapy" - Pharmac. Therap. 27 (1985) 333.

G. Gorneva, J. Mladenova, S. Zakhariev, S. Stoev, B. Alexiev, A. Spassov, M. Karaivanova, E. Golovinsky - "Di-(2-halogenethyl)hydrazides of Amino Acids,  their Analogs and Derivatives: Antitumor Activity, Effect on DNA, RNA, Prorein Synthesis and Cell Cycle Progression" - CMEA Chemotherapy Symposium 1984; S. Ekhard and S. Kerpel-Fronius, Edt.; Akad. Kiado, Budapest 1985.

K. Grancharov, G.-J. Krauss, N. Spassovska, J. Miersch, L. Maneva, J. Mladenova, E. Golovinsky - "Inhibitory effect of pyruvic acid semi- and thiosemicarbazones on the growth of bacteria, yeasts, experimental tumors and plant cells" - Pharmazie 40 (1985) 574.

G.-J. Krauss,  J. Miersch, K. Grancharov, F. Bublitz, N. Spassovska, E. Golovinsky - "The Effect of Pyruvic Acid Thiosemicarbazone on Ornitine Carbamoil Transferase of Lycopersicol esculentum Mill" - Biologia Plantarum (Praha) 28 (3), (1986) 174.

R. Natcheva, I. Manolov, E. Golovinsky - "Kinetics of the Intramolecular Cyclization of Bis (2-chloroethyl)aminoethyl Esters of Carboxylic Acids" - Die Pharmazie 41 (1986) 642.

K. Grancharov, G. Gorneva, I. Mladenova, K. Norpoth, E. Golovinsky - "Lack of Genotoxic and Cytostatic effects of the Herbicide Lenacil on Mouse Tumor Cells and on some Salmonella typhimurium Strains" - Arzneimittel-Forschung 36 (II), (11), (1986) 1660-1663.

I. Kostova, N. Spassovska, L. Maneva, E. Golovinsky, I. Ognyanov - "Reaction of Retenoids with Hydrazine" - Heterocycles 24 (9), (1986) 2471-2477.

K. Nikolova, L. Maneva, G. Karamanov, E. Golovinsky - "Studies on the Antimycotic Activity of 5-Fluoroorotic Acid" - Methods and Findings in Experim. and Clinical Pharmacology 9 (2), (1987) 85-89.

J. Miersch, K. Grancharov, G.-J. Krauss, N. Spassovska, L. Maneva, I. Mladenova, E. Golovinsky - "Biological Activity and Mode of Action of some Dihydroorotic and Dihydroazaorotic Acid Derivatives" - Biomed. Biochim. Acta 46 (5), (1987) 307-315.

G. Schuster, Ch. Aristoph, E. Golovinsky - "Analogues of Pyrimidine Base Precursors as Antiphytoviral Agents" - Antiviral Research 7 (1987) 179-184.

L. Maneva, S. Zakhariev, S. Stoev, E. Golovinsky - "Sulfoanalogs of Asparagine and Gentamine - Synthesis and Antibacterial Activity" In: "Molecular and Cellular Regulation of Enzyme Activity, C. Wasternack, A. Barth (Eds.), Martin-Luther-Universitat Halle (Saale) 1987, pp. 40-44.

C. Verkoyen, E. Golovinsky, G. Muller, M. Kolbel, K. Norpoth - "Synthese von 7-Phenylguanin und 2-substituierten 7-Arylhypoxanthinen" - Liebigs Annalen d. Chemie 1987, 957-960.

W. Stucker, E. Golovinsky, G. Muller, M. Oberst, K. Maher, K. Norpoth - "New Color Reagrnts for the Analysis of Alkylating Agents" - Fresenius Zeitschr. Anal Chem. 330, (1988) 42-45.

I. Manolov, E. Golovinsky - "Attempt to Estabish a Correlation between the Acylation Ability and Antitumor Activity of some Bis(2-chloroethyl)aminoethyl Esters of Carboxylic Acids" - Die Pharmazie 43 (1988) 218-219.

K. Halacheva, Z. Zhelev, T.  Pajpanova, A. Hubenova, M. Spassova, Ch. lexiev, E. Golovinsky - "Lysine-Orotate Potentiate the Toxicity of an Extract of the Mushroom Amanita Phalloides" - Toxicon 26 (6), (1988) 571-576.

S. Stoev, S. Zakhariev, E. Golovinsky, H.-G. Gattner, V. Naithani, A. Wollmer, D. Brandenburg - "Synthesis and Properties of [A19-(p-Fluoropheylalanine)]Insulin" - Biol. Chem. Hoppe-Seyler 369 (1988) 1307-1315.

S. Zakhariev, G. Videnov, S. Stoev, E. Golovinsky - "Asymmetrical Derivatives of Diaminosuberic Acid Useful in Peptide Synthesis" - Peptides 1988, 307-309.

S. Lozeva, S. Zakhariev, S. Stoev, S. Taksirov, E. Golovinsky - "Synthese von N,N-Di(2-Bromoethyl)hydraziden einiger Naturlichen L-Aminosauren" - Pharmazie 44 (5), (1989). 316-317.

T. Pajpanova, S. Stoev, J. Miersch, G.-J. Krauss, E. Golovinsky - "Canavanine Derivatives: Synthesis and Application" - Conf. Proc. 5th Intern. Conf. Chem. Biothech. Biol. Active Natural Prod., BAS - Sofia, 1989.

R. Gugova, S. Taksirov, G. Demirov, E. Golovonsky - "N-Arylacylnitrososemicarbazides: Synthesiss and in vivo Activity against L1210" - Conf. Proc. 5th Intern. Conf. Chem. Biotechnol. Biol. Active Natural Products, BAS - Sofia, 1989.

S. Zakhariev, S. Stoev, B. Alexiev, L. Maneva, E. Golovinsky - "Synthese und Geschwulsthemmende Wirkung in vivo von N,N-Di(2-chlorethyl)hydraziden naturlicher L-Aminocarbonsauren" - Pharmazie 44 (9), (1989) 608-611.

S. Zakhariev, S. Stoev, K. Maneva, M. Ilarionova, D. Todorov, E. Golovinsky - "Synthesis and antirumor effect of N₁-acyl derivatives of 1-cystine-bis[N,N-di(2-chloroethyl)]dihydrazide" - Pharmazie 44 (11), (1989) 763-765.

L. Jossifova, I. Manolov, E. Golovinsky - "Antibakterielle Wirkung einiger gesattigter und ungesattigter langkettiger Carbonsauren und deren Bis(2-chlorethyl)aminoethylester in vitro" - Pharmazie 44 (12), (1989) 854.

I. Pajeva, I. Manolov, E. Golovinsky - "Structure - activity relationship investigation of bis(2-chloroethyl)aminoethylesters of some carboxilic acids". Pharmazie 45 (1990) 361-365.

I. Pajeva, E. Golovinsky - "Substructural Analysis of Antineoplastic Compounds in Respect of in vivo Tumor Models" - Struct.-Activ. Relat. 9 (1990) 216-222.

E. Golovinsky, R. Gugova, K. Norpoth, E. Mohtashamipur - "Mutagenic activity of some newly synthesized cytostatic 1-(2-chloroethyl)-4-aryacyl-1-nitrososemicarbazides in the Salmonella/ mammalian microsome assay". J. Cancer Res. Clin. Oncol. 117, (1990) 1-3.

S. Zakhariev, E. Golovinsky, S. Stoev, L. Maneva, B. Alexiev - "Synthese und geschwulsthemmende Wirkung von N,N-Di-(2-chlorethyl)-hydrazinen der alfa-Aminocarbonsaureantimetabolite". Pharmazie 44 (1989) 541-544.

K. Grancharov, J. Mladenova, E. Golovinsky - "Inhibition of uridine phosphorylase by some pyrimidine derivatives". Biochem. Pharmacol. 41 (11), (1991) 1769-1772.

D. Lazarov, E. Golovinsky - "The Integrated course NATURE in the Curricular struture of BARGEP". Science and technology education, Document series UNESCO, No 38, (1990) p.p. 50-51.

E. Karanov, V. Alexieva, E. Golovinsky, M. Haimova - "Cytokinin and anticytokynin activity of some 4-substituted 1H-pyrazoles and 8-aza analogues of adenine”. Plant-Growth regulation 13 (1992) 7-11.

R. Gugova, A. Papageorgiu, S. Taxirov, V. Topacbashian, E. Margariti, L. Boutis, D. Mourelatos, T. Dozi-Vassiliades, E. Golovinsky, G. Demirov - "4-Aroyl-1-nitrosohydrazinesemicarbazides: synthesis, in vivo and in vitro antitumor activity". Europ. J. Med. Chemistry 27 (1992) 745-750.

D. Sidzhakova, B. Panajotova, Z. Mardirossjan, S. Tabakova, L. Maneva, V. Marinova, E. Golovinsky - "Synthesis and biological activity of mono- and bishydrazones of cyclic aminoguanidines". Pharmazie 48 (6), (1993) 417-419.

E. Golovinsky - "Der Krebs- eine Herausforderung fur die Chemotherapie". Chemie in Labor und Biothechnik 44 (7), (1993) 341-346.

J. Miersch, T. Pajpanova, K. Grancharov, G.-J. Krauss, H. Tintemann, E. Golovinsky - "Some new canavanine derivatives: synthesis and biological activity". Aminoacids 5 (1), (1993) 126.

M. Shopova, S. Tabacova, S. Taxirov, E. Golovinsky - "Synthesis and biological activity of some N₁-substituted orotic acids". Pharmazie 48 (1993) 861.

M. Somleva, M. Odjakova, E. Golovinsky - "In vitro effect of some pyrimidine analogues on embriogenic response of Dactylis-glomerata leaf eklants". J. Plant Physiology 142 (1993) 765-767.

Z. Mincheva, V. Kalcheva, E. Golovinsky, S. Tabacova - "Synthesis and in vitro activity of new cephem derivatives with benzoxalons ring". Pharmazie 48 (11), (1993) 859-860.

A. Bocheva, D. Getova, T. Pajpanova, N. Stoeva, S. Stoev, E. Golovinsky - "Central and Peripheral Effects of Some Newly Synthetized Enkephalines". Neuropeptides 26 (1994) 41.

C. Schell, O. Lantermann, W. Popp, .Varenholtz, J. Thomale, R. Gugova, E. Golovinsky, K. Norpoth - "Genotoxic and cytotoxic effects of 4-aroyl-1-nitrosohydrazinecarboxamides on O6-alkylguanine-DNA-alkyltransferase-positive and -negative human cell lines". J. Cancer Res. Clin. Oncol. 120 (1994) 403-408.

M. Somleva, V. Kapchina, V. Alexieva, E. Golovinsky - "Anticytokinin efffects on in vitro response of embriogenic and nonembrinogenic genotypes of Dactylis glomerata L.". Plant Growth Regulation 16 (1995) 109-112.

V. Alexieva, I. Sergiev, E. Karanov, E. Golovinsky, E. Stanoeva, M. Haimova, G. Petrov - "Anticytokinin activity of 4-substituted triazolo[4,5-d]pyrimidines". J. Plant Growth Regulation 13 (1994) 123-129.

T. Pajpanova, S. Stoev, E. Golovinsky, G.-J. Krauss, J. Miersch - "Canavanine useful in peptide synthesys". Amino Acids (1996) in press.

B. Nesterova, T. Pajpanova, S. Simova, S. Tabakova, E. Golovinsky, M. Haimova - "Synthesis and Antibacterial Activity of 7 β-{3(Un)substituted-2-aminopropionamido}-3-vinylcephalosporins and related Compounds". Arch. Pharm. (Weinheim) 328 (1995) 1.

J. Miersch, K. Grancharov, T. Pajpanova, R. Baumbach, S. Tabakova, S. Stoev, G.-J. Krauss, E. Golovinsky - "Ecological significance of Canavanine and biological activity of some canavanine derivatives". In: Guanidino Compounds in Biology and Medicine; P. deDeyn, B. Marescan, V. Stalon and I. Qureshi (Eds.), Publ. J. Libbey, Montreal, 1995.

Z. Naydenova, K. Grancharov, M. Shopova, E. Golovinsky - "Inhibition of UDP-glucoronyltransferase activity in rat liver microsomes by pyridimidine derivatives". Comp. Biochem. Physiol. 112c, n 3, (1995) 1-5.

Z. Naydenova, Z. Urshev, E. Golovinsky, K.  Grancharov - "Influence of Pesticides on UDP-glucoronosyltransferase in Rat Liver Microsomes". Pestic. Sci. (1996) 43.

A.Bocheva, T. Pajpanova, E. Golovinsky, M. Lazarova-Bakarova - "Studies on pain modulation by newly-synthesized analogues of kyotorphin". Proc. 7th International Sympozium "The Pain Clinic", Monduzzi Editore, Bologna, 1996, p.p.15-18.

I. Stankova, G. Videnov, A. Galabov, E. Golovinnsky - "Amino Acid and peptide derivatives of 5-Bromo-2'-deoxiuridine (BrdUrd): Synthesis, characterisation and biological activity". Peptides, 1996.

Z. Naydenova, D. Alargov, K. Grancharov, E. Golovinsky - "Inhibitory Effects of 5'-O-Amino-Acid Derivatives of Uridine on UDP-glucuronosyltransferase in Rat Liver Microsomes". Exp. Toxic. Pathol. 48 (1996) Suppl. II. 295-298.

R. Gugova, V. Topakbashian, S. Lozeva, S. Dimov, E. Golovinsky - "Synthesis and Antitumour Activity of several New 4-Aroyl-1-nitrosohydrazinecarboxamides". Drugs Under Exper. Clin. Res. 23 (1997) 71-75.

D. Alargov, Z. Naydenova, K. Grancharov, P. Denkova, E. Golovinsky - "Synthesis of Some 5'-O- Amino Acid Derivatives of Uridine as Potential Inhibitors of UDP-glucuronosyltransferase". Monatshefte f. Chemie 128 (1997) 725-732.

D. K. Alargov, P.S. Denkova, E. V. Golovinsky - "Glucuronidation of Serine and Threonine". Monatshefte f. Chemie 128 (1997) 733-736.

L. Staleva, L. Waltscheva, E. Golovinsky, P. Venkov - "Enhanced cell permeability increases the sensitivity of a yeast test for mutagens". Mutation Research 370 (1996) 81-89.

M. Stanchev, A. Bocheva, S. Todorov, E. Golovinsky - “Effects of newly synthesized amino acids containing thiazole residues on electrically avoced smooth muscle contractions”. Meth. Find. Exp. Clin. Pharmacol. 20 (1998) 171-177.

Z. Naydenova, K. Grancharov, D. Alargov, E. Golovinsky, I. Stanoeva, L. Shalamanova, I. Pajeva - “Inhibition of UDP-glucuronosyltransferase by 5’-amino-Acid and oligopeptide derivatives of uridine: structure - activity relationships”. Z. Naturforschg. 53c (1998) 173-181.

T. Pajpanova, K. Grancharov, E. Golovinsky, L. Kazakov, J. Miersch, G.-J. Krauss – “Amino Acid and Peptide Analogues of Non-protein Amino Acid Canavasnine: Synthesis and Biological Activity”. Peptides 1996, R. Ramage and E. Epton (Eds.), EPS, 1998, pp. 705-706.

D. Alargov, Z. Naydenova, K. Grancharov, P. Denkova, E. Golovinsky – “Synthesis of 5’-O-Oligopeptide Derivatives of Uridine as Inhibitors of UDP-Glucuronosyltransferase”. Monatshefte f. Chemie, 129 (1998) 755-760.

S. Tabakova, I. Manolov, T. Kantardjiev, G. Mateev, K. Stoichkov, A. Braikova, V. Vakhan, E. Golovinsky – “Anticandidial Effect of Phenylbutene Derivatives and Their Interaction with Ergosterol”. Z. Naturschg. (1998).

I. Stankova, M. Simeonov, V. Maximova, A. Galabov, E. Golovinsky – “Synthesis and Anti-Virus Activity of Some Nucleosides Analogues”. Z. Naturforschg, 54c (1999) 75-83.

E. Golovinsky, Z. Naydenova, K. Grancharov – “UDP-Glucuronosyltransferase inhibitors”. Europ. J. Drug Metabol. Pharmacokinetics. 23, No 4, (1998) 453-456.

D. Alargov, R. Gougova, P. Denkova, G. Müller, E. Golovinsky – “Synthesis of Cyclohexane Containing 5’-O-Glycine Derivatives of Uridine as Potential Inhibitors of UDP-glucuronosyltransferase”. Monatshefte f. Chemie, 130 (1999) 937-943.

I. Stankova, G. Videnov, S. Tabakova, E. Golovinsky, G. Jung – “Synthesis of Novel Imidazole, Thiazole, Oxazole Substituted Peptides, Cyclotetrapeptide and their Antibacterial Activity in vitro”. Peptides 1988, pp 248-249. Acad. Kiado Budapest, S. Bajusz and F. Hudecz (Eds.).

Z. Naydenova, G.-J. Krauss, E. Golovinsky, K. Grancharov – “Effect of s-triazine and phenoxyalkanoic acid herbicides on UDP-glucuronosyltransferase rat liver microsomes”. Pestic. Sci. 55 (1999) 825-830.

M. Stanchev, S. Tabakova, G. Videnov, E. Golovinsky, G. Jung – “Synthesis and Antimicrobial Activity in vitro of New Amino Acids and Peptides Containing Thiazole and Oxazole Moieties”. – Arch. Pharm. Pharm. Med. Chem. 332 (1999) 297-304.

I. Stankova, G. Videnov, E. Golovinsky, G. Jung – “Synthesis of Thiazole, Imidazole, and Oxazole Containing Amino Acids for Peptide Backbone Modification”. J. Peptide Sci. 5 (1999) 392-398.

A. Bocheva, R. Zamfirova, T. Pajpanova, S. Todorov, M. Georgieva, E. Golovinsky – “Effect of Di-phenylhydranine on the Tyr-Mif-1 Antinociception in Rats”. Arch. Physiol. Biochem. 106, No.5, (1998) 378-383.

T. Pajpanova, A. Bocheva, E. Golovinsky – “Effects of Newly Synthesized Analogs of MIF-1 Containing Unnatural Amino Acids on Electrically Evoced Smeooth Muscle Contractions”. Methods Find. Exp. Clin. Pharmacol. 21 (9), (1999) 591-594.

M. Stanchev, T. Pajpanova, E. Golovinsky – “Synthesis and antibacterial activity of some new non-proteinogenic amino acids containing thiazole residues”. Amino Acids 18 (2000) 177-191.

Zh. Velkov, R. Pelova, St. Stoev, E. Golovinsky “Synthesis and characterization of some Pt(II) and Pt(II) Complexes with Thioamide Analogues of Amino Acids”. J. Coord. Chem. 26 (1992) 75-78.

K. Grancharov, Z. Naydenova, S. Lozeva, E. Golovinsky – “Natural and synthetic inhibitors of UDP-glucuronosy;transferase”. Parmac. Therap. 89 (2001) 1-16.

I. G. Stankova, D. A. Beschkov, E. V. Golovinsky – “Synthesis and in vitro Evaluation for Anti-HIV Effect and Toxicity of a New Peptides Analogues of 3’-Azido-3’-deoxythymidine”. Peptides 2000, J. Martinez and J.-Alain Fehrentz (Eds.), EDK, Paris, France (2001) p.p. 745-746.

K. Grancharov, H. Engelberg, Z. Naydenova, G. Müller, A.W. Rettenmeier, E. Golovinsky – “Inhibition of UDP-glucuronosyltransferases in rat liver microsomes by natural mutagens and carcinogens”. Arch. Toxicol. 75 (2001) 609-612.

J. Miersch, K. Grancharov, T. Pajpanova, S. Tabakova, S. Stoev, G.-J. Krauss, E. Golovinsky – “Synthesis and biological activity of canavanine hydrazide derivatives”. Amino Acids, 18 (2000) 41-59.

D. Kushev, R. Grünert, N. Spassovska, E. Golovinsky, P. Bednarski – “Unusual reactivity of cytotoxic cis-dihydrazide Pt (II) complexes in aqueous solutions”. J. Inorganic. Biochem. 96, No 4, (2003) 469-477.

T. Dzimbova, T. Pajpanova, E. Golovinsky – “Synthesis of some sulfoguanidino group-containing amino acids”. Collection Symposium Letters 6 (2003) 12-14.

I. G. Stankova, D. A. Beschkov, E. V. Golovinsky – “Synthesis and in vitro Evaluation for Anti-HIV Effect and Toxicity of a New Peptides Analogues of 3’-Azido-3’-deoxythymidine”. Peptides 2000, J. Martinez and J.-Alain Fehrentz (Eds.), EDK, Paris, France (2001) p.p. 745-746.

K. Grancharov, H. Engelberg, Z. Naydenova, G. Müller, A.W. Rettenmeier, E. Golovinsky – “Inhibition of UDP-glucuronosyltransferases in rat liver microsomes by natural mutagens and carcinogens”. Arch. Toxicol. 75 (2001) 609-612.

K. Grancharov, E. Golovinsky – “Uridine Phosphorilase Inhibitors: Structure-Activity Relationships”. C. r. Acad. Bulgare Sci. 55, No 12, (2002) 79-82.

J. Miersch, K. Grancharov, T. Pajpanova, S. Tabakova, S. Stoev, G.-J. Krauss, E. Golovinsky – “Synthesis and biological activity of canavanine hydrazide derivatives”. Amino Acids 18 (2000) 41-59.

G. Gorneva, E. Golovinsky – “Comparative Study of the Appoptogenic Effect of Fluoropyrimidines on Marine Leukemia Cells”. Nova Acta Leopoldina, NF 87, No 329, (2003).183-189.

G. Satchanska, E. Golovinsky, S. Selenska-Pobell – “Bacterial diversity in a sil sample from uranium mining waste pile as estimated via a culture-independent 16S rRNA approach” C. r. Acad. Bulgare Sci., 57,No 4, (2004) 75 – 82.

M. Pesheva, K. Antonios, T. Pajpanova, E. Golovinsky – “Inhibition of the activity of yeast enzyme invertase by the arginine antimetabolite L-canavanine”. C. r. Acad. Bulgare Sci., 56 No 11, (2003) 55 – 58.

T. Pajpanova, A. Bocheva, L. Kazakov, E. Golovinsky – “Synthrsis and comparative study of opioid effects of canavanine analogs of Leu-enkefalin and dalargin” – C. r. Acad. Bulgare Sci. 57 No 3, (2004) 39 – 44.

M. Stanchev, A. Bocheva, T. Angelov, S. Todorov, T. Pajpanova, E. Golovinsky – “Structure-Activity Studies of Peptidomimetics Containing Azole Residues. Effects of Cholinergic Neurotransmission”. Bulg. Chem. Commun. 33, (2001) 65 – 72.